Skip to main navigation Skip to search Skip to main content

Three stories on Eph kinase inhibitors: From in silico discovery to in vivo validation

  • A Unzue
  • , K Lafleur
  • , HT Zhao
  • , T Zhou
  • , J Dong
  • , P Kolb
  • , Johanna Liebl
  • , S Zahler
  • , A Caflisch
  • , C Nevado

    Research output: Contribution to journalReview articlepeer-review

    26 Citations (Web of Science)
    Original languageEnglish
    Pages (from-to)347-366
    JournalEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
    Volume112
    DOIs
    Publication statusPublished - 2016

    Keywords

    • STRUCTURE-BASED DESIGN
    • RECEPTOR TYROSINE KINASES
    • FRAGMENT-BASED DOCKING
    • GROWTH-FACTOR RECEPTOR
    • PROTEIN-KINASES
    • BREAST-CANCER
    • TUMOR-GROWTH
    • MAP KINASE
    • BIOLOGICAL SIGNIFICANCE
    • MOLECULAR-DYNAMICS

    Cite this