Three stories on Eph kinase inhibitors: From in silico discovery to in vivo validation

A Unzue, K Lafleur, HT Zhao, T Zhou, J Dong, P Kolb, Johanna Liebl, S Zahler, A Caflisch, C Nevado

    Research output: Contribution to journalReview articlepeer-review

    25 Citations (Web of Science)
    Original languageEnglish
    Pages (from-to)347-366
    JournalEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
    Volume112
    DOIs
    Publication statusPublished - 2016

    Keywords

    • STRUCTURE-BASED DESIGN
    • RECEPTOR TYROSINE KINASES
    • FRAGMENT-BASED DOCKING
    • GROWTH-FACTOR RECEPTOR
    • PROTEIN-KINASES
    • BREAST-CANCER
    • TUMOR-GROWTH
    • MAP KINASE
    • BIOLOGICAL SIGNIFICANCE
    • MOLECULAR-DYNAMICS

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