Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core.

Miroslav Sisa; Marcela Dvorakova; Veronika Temml; Veronika Jarosova; Tomas Vanek; Premysl Landa

doi:10.1016/j.ejmech.2020.112620

Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core.

Miroslav Sisa
, Marcela Dvorakova
, Veronika Temml (Co-author)
, Veronika Jarosova
, Tomas Vanek
, Premysl Landa

Insitute of Pharmacy

Research output: Contribution to journal › Original Article › peer-review

11 Citations (Web of Science)

Original language	English
Pages (from-to)	112620
Journal	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume	204
DOIs	https://doi.org/10.1016/j.ejmech.2020.112620
Publication status	Published - 2020

Keywords

SELECTIVE-INHIBITION
5-LIPOXYGENASE
CYCLOOXYGENASE
DERIVATIVES

Access to Document

10.1016/j.ejmech.2020.112620

Cite this

Sisa, M., Dvorakova, M., Temml, V., Jarosova, V., Vanek, T., & Landa, P. (2020). Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY , 204, 112620. https://doi.org/10.1016/j.ejmech.2020.112620

Sisa, Miroslav ; Dvorakova, Marcela ; Temml, Veronika et al. / Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core. In: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 2020 ; Vol. 204. pp. 112620.

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title = "Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core.",

keywords = "SELECTIVE-INHIBITION, 5-LIPOXYGENASE, CYCLOOXYGENASE, DERIVATIVES",

author = "Miroslav Sisa and Marcela Dvorakova and Veronika Temml and Veronika Jarosova and Tomas Vanek and Premysl Landa",

year = "2020",

doi = "10.1016/j.ejmech.2020.112620",

language = "English",

volume = "204",

pages = "112620",

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Sisa, M, Dvorakova, M, Temml, V, Jarosova, V, Vanek, T & Landa, P 2020, 'Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core.', EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY , vol. 204, pp. 112620. https://doi.org/10.1016/j.ejmech.2020.112620

Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core. / Sisa, Miroslav; Dvorakova, Marcela; Temml, Veronika (Co-author) et al.
In: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY , Vol. 204, 2020, p. 112620.

Research output: Contribution to journal › Original Article › peer-review

TY - JOUR

T1 - Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core.

AU - Sisa, Miroslav

AU - Dvorakova, Marcela

AU - Temml, Veronika

AU - Jarosova, Veronika

AU - Vanek, Tomas

AU - Landa, Premysl

PY - 2020

Y1 - 2020

KW - SELECTIVE-INHIBITION

KW - 5-LIPOXYGENASE

KW - CYCLOOXYGENASE

KW - DERIVATIVES

U2 - 10.1016/j.ejmech.2020.112620

DO - 10.1016/j.ejmech.2020.112620

M3 - Original Article

C2 - 32738413

SN - 0223-5234

VL - 204

SP - 112620

JO - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

JF - EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

ER -

Sisa M, Dvorakova M, Temml V, Jarosova V, Vanek T, Landa P. Synthesis, inhibitory activity and in silico docking of dual COX/5-LOX inhibitors with quinone and resorcinol core. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY . 2020;204:112620. doi: 10.1016/j.ejmech.2020.112620