Steroid sulfatase inhibiting lanostane triterpenes - Structure activity relationship and in silico insights.

Ulrike Grienke; Teresa Kaserer; Benjamin Kirchweger; George Lambrinidis; Ralph T Kandel; Paul A Foster; Daniela Brigitte Schuster; Emmanuel Mikros; Judith M Rollinger

doi:10.1016/j.bioorg.2019.103495

Steroid sulfatase inhibiting lanostane triterpenes - Structure activity relationship and in silico insights.

Ulrike Grienke, Teresa Kaserer, Benjamin Kirchweger, George Lambrinidis, Ralph T Kandel, Paul A Foster, Daniela Brigitte Schuster (Co-author), Emmanuel Mikros, Judith M Rollinger

Insitute of Pharmacy

Research output: Contribution to journal › Original Article › peer-review

11 Citations (Web of Science)

Original language	English
Pages (from-to)	103495
Journal	BIOORGANIC CHEMISTRY
Volume	95
DOIs	https://doi.org/10.1016/j.bioorg.2019.103495
Publication status	Published - 2020

Keywords

POTENT INHIBITORS
REVERSIBLE INHIBITORS
ESTRONE SULFATASE
IROSUSTAT
PROTEIN
PHARMACOPHORE
DISCOVERY

Access to Document

10.1016/j.bioorg.2019.103495

Cite this

@article{aa4a4fef74574f64a334e33cdd5cfb99,

title = "Steroid sulfatase inhibiting lanostane triterpenes - Structure activity relationship and in silico insights.",

keywords = "POTENT INHIBITORS, REVERSIBLE INHIBITORS, ESTRONE SULFATASE, IROSUSTAT, PROTEIN, PHARMACOPHORE, DISCOVERY",

author = "Ulrike Grienke and Teresa Kaserer and Benjamin Kirchweger and George Lambrinidis and Kandel, {Ralph T} and Foster, {Paul A} and Schuster, {Daniela Brigitte} and Emmanuel Mikros and Rollinger, {Judith M}",

note = "Schuster: Paracelsus Med Univ Salzburg, Dept Pharmaceut *** Med Chem, Inst Pharm, Salzburg, Austria",

year = "2020",

doi = "10.1016/j.bioorg.2019.103495",

language = "English",

volume = "95",

pages = "103495",

journal = "BIOORGANIC CHEMISTRY",

issn = "0045-2068",

}

TY - JOUR

T1 - Steroid sulfatase inhibiting lanostane triterpenes - Structure activity relationship and in silico insights.

AU - Grienke, Ulrike

AU - Kaserer, Teresa

AU - Kirchweger, Benjamin

AU - Lambrinidis, George

AU - Kandel, Ralph T

AU - Foster, Paul A

AU - Schuster, Daniela Brigitte

AU - Mikros, Emmanuel

AU - Rollinger, Judith M

N1 - Schuster: Paracelsus Med Univ Salzburg, Dept Pharmaceut *** Med Chem, Inst Pharm, Salzburg, Austria

PY - 2020

Y1 - 2020

KW - POTENT INHIBITORS

KW - REVERSIBLE INHIBITORS

KW - ESTRONE SULFATASE

KW - IROSUSTAT

KW - PROTEIN

KW - PHARMACOPHORE

KW - DISCOVERY

U2 - 10.1016/j.bioorg.2019.103495

DO - 10.1016/j.bioorg.2019.103495

M3 - Original Article

C2 - 31855822

SN - 0045-2068

VL - 95

SP - 103495

JO - BIOORGANIC CHEMISTRY

JF - BIOORGANIC CHEMISTRY

ER -