Pharmacophore-based discovery of FXR agonists. Part I: Model development and experimental validation.

Daniela Brigitte Schuster, Patrick Markt, Ulrike Grienke, Judit Mihaly-Bison, Markus Binder, Stefan M Noha, Judith M Rollinger, Hermann Stuppner, Valery N Bochkov, Gerhard Wolber

    Research output: Contribution to journalOriginal Articlepeer-review

    31 Citations (Web of Science)
    Original languageEnglish
    Pages (from-to)7168-7180
    JournalBIOORGANIC & MEDICINAL CHEMISTRY
    Volume19
    Issue number23
    DOIs
    Publication statusPublished - 2011

    Keywords

    • FARNESOID-X-RECEPTOR
    • BILE-ACID RECEPTOR
    • NUCLEAR RECEPTOR
    • DRUG DISCOVERY
    • POTENT
    • IDENTIFICATION
    • ANTAGONIST
    • ACTIVATION
    • DATABASE
    • ANALOGS

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